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4-[1-[4-[2-(dimethylamino)ethoxy]phenyl]-2-phenylbut-1-enyl]phenol and diethylstilbestrol

4-[1-[4-[2-(dimethylamino)ethoxy]phenyl]-2-phenylbut-1-enyl]phenol has been researched along with diethylstilbestrol in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (25.00)18.2507
2000's5 (62.50)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fine, RL; Rao, US; Scarborough, GA1
Bélanger, A; Caron, B; Cloutier, J; Dory, YL; Favre, A; Gauthier, S; Labrie, C; Labrie, F; Larouche, D; Leblanc, G; Mailhot, J; Martel, C; Mérand, Y; Ouellet, C; Schwerdtfeger, A; Simard, J1
Strassburg, CP; Tukey, RH1
Dunn-Dufault, R; Feher, M; Kalbakji, A; Mercure, J; Pagé, M; Peter, MG; Redden, PR; Schmidt, JM; Tremblay, GB1
Chao, EY; Collins, JL; Gaillard, S; Jones, DG; McDonnell, DP; Miller, AB; Orband-Miller, LA; Shearer, BG; Willson, TM; Zuercher, WJ1
Ernst, B; Lill, MA; Vedani, A; Winiger, F1
Armstrong, MD; Arteaga, CL; Brown, HA; Buck, JR; Cho, HP; Criswell, TL; Lindsley, CW; Scott, SA; Selvy, PE; Thomas, AL1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1

Reviews

1 review(s) available for 4-[1-[4-[2-(dimethylamino)ethoxy]phenyl]-2-phenylbut-1-enyl]phenol and diethylstilbestrol

ArticleYear
Human UDP-glucuronosyltransferases: metabolism, expression, and disease.
    Annual review of pharmacology and toxicology, 2000, Volume: 40

    Topics: Autoimmunity; Chromosome Mapping; Glucuronides; Glucuronosyltransferase; Humans; Hyperbilirubinemia; Neoplasms; Steroids; Terminology as Topic

2000

Other Studies

7 other study(ies) available for 4-[1-[4-[2-(dimethylamino)ethoxy]phenyl]-2-phenylbut-1-enyl]phenol and diethylstilbestrol

ArticleYear
Antiestrogens and steroid hormones: substrates of the human P-glycoprotein.
    Biochemical pharmacology, 1994, Jul-19, Volume: 48, Issue:2

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Cells, Cultured; Estradiol; Estrogen Antagonists; Humans; Hydrocortisone; Insecta; Membrane Glycoproteins; Progesterone; Steroids; Transfection; Verapamil

1994
(S)-(+)-4-[7-(2,2-dimethyl-1-oxopropoxy)-4-methyl-2-[4-[2-(1-piperidinyl)-ethoxy]phenyl]-2H-1-benzopyran-3-yl]-phenyl 2,2-dimethylpropanoate (EM-800): a highly potent, specific, and orally active nonsteroidal antiestrogen.
    Journal of medicinal chemistry, 1997, Jul-04, Volume: 40, Issue:14

    Topics: Administration, Oral; Animals; Benzopyrans; Binding, Competitive; Breast Neoplasms; Cytosol; Diethylstilbestrol; Estradiol; Estrogen Antagonists; Female; Humans; Mice; Molecular Structure; Ovariectomy; Piperidines; Propionates; Raloxifene Hydrochloride; Receptors, Estrogen; Stereoisomerism; Structure-Activity Relationship; Uterus

1997
De novo design, synthesis, and evaluation of novel nonsteroidal phenanthrene ligands for the estrogen receptor.
    Journal of medicinal chemistry, 2003, Apr-10, Volume: 46, Issue:8

    Topics: Animals; Binding, Competitive; Cell Division; Cell Line; Chlorocebus aethiops; Computer Simulation; Estrogen Receptor alpha; Estrogen Receptor beta; Estrogen Receptor Modulators; Humans; Ligands; Models, Molecular; Phenanthrenes; Radioligand Assay; Receptors, Estrogen; Structure-Activity Relationship; Transcription, Genetic; Tumor Cells, Cultured

2003
Identification and structure-activity relationship of phenolic acyl hydrazones as selective agonists for the estrogen-related orphan nuclear receptors ERRbeta and ERRgamma.
    Journal of medicinal chemistry, 2005, May-05, Volume: 48, Issue:9

    Topics: Binding, Competitive; Estrogen Receptor beta; Fluorescence Resonance Energy Transfer; Genes, Reporter; Heat-Shock Proteins; HeLa Cells; Humans; Hydrazines; Ligands; Molecular Mimicry; Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha; Phenols; Receptors, Estrogen; Structure-Activity Relationship; Transcription Factors

2005
Impact of induced fit on ligand binding to the androgen receptor: a multidimensional QSAR study to predict endocrine-disrupting effects of environmental chemicals.
    Journal of medicinal chemistry, 2005, Sep-08, Volume: 48, Issue:18

    Topics: Benzhydryl Compounds; Binding Sites; Diethylstilbestrol; Endocrine System; Hydrocarbons, Chlorinated; Ligands; Models, Molecular; Molecular Conformation; Phenols; Phytoestrogens; Quantitative Structure-Activity Relationship; Receptors, Androgen; Testosterone; Thermodynamics; Xenobiotics

2005
Design of isoform-selective phospholipase D inhibitors that modulate cancer cell invasiveness.
    Nature chemical biology, 2009, Volume: 5, Issue:2

    Topics: Breast Neoplasms; Drug Design; Enzyme Inhibitors; Humans; Isoenzymes; Neoplasm Invasiveness; Phospholipase D

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010